Print version: Silverman, Richard B. Organic chemistry of drug design and drug action. Third edition. Amsterdam : Elsevier, c2014 xviii, 517 pages ISBN 9780123820303
Introduction -- Lead discovery and lead modification -- Receptors -- Enzymes -- Enzyme inhibition and inactivation -- Dna-interactive agents -- Drug resistance and drug synergism -- Drug metabolism -- Prodrugs and drug delivery systems.